產(chǎn)品名稱 CP 100356 hydrochloride from TOCRIS BIOSCIENCE
    產(chǎn)品貨號 4193/10
    產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
    產(chǎn)品規(guī)格 10 mg
    產(chǎn)品品牌 TOCRIS BIOSCIENCE
    產(chǎn)品概述
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    Product NameCP 100356 hydrochloride
    DescriptionHigh affinity P-glycoprotein (P-gp) inhibitor (Ki values are 58 and 94 nM for mouse Pgp1a and Pgp1b isoforms). Inhibits calcein-AM uptake in MDR1-transfected MDCKII cells (IC50 = 0.5 μM) and prazosin transport in BCRP-transfected MDCKII cells (IC50 = 1.5 μM). Displays weak or no inhibitory activity against MRP1, OATP1B1 and several major human P450 enzymes (IC50 > 50 μM). Purity 98%. MW (observed): 597.1
    Size10 mg
    Concentrationn/a
    Applicationsn/a
    Other Names4-(3,4-Dihydro-6,7-dimethoxy-2(1H)-isoquinolinyl)-N-2[2-(3,4-dimethoxyphenyl)ethyl]-6,7-dimethoxy-2-quinazolinamine hydrochloride
    Gene, Accession, CAS #CAS: 142715-48-8
    Catalog #4193/10
    Price
    Order / More InfoCP 100356 hydrochloride from TOCRIS BIOSCIENCE
    Product Specific ReferencesPubMed: 26046259
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