A cannabimimetic with a relatively low-affinity for the CB1 receptor (Ki = 855 nM); interferes with the action of the potent CB1 agonist WIN 55,212-2, suggesting that it acts as a silent CB1 antagonist; reduces food intake and body weight gain in obese Zucker rats
Size
10 mg
Concentration
n/a
Applications
n/a
Other Names
cannabimimetic CBs cannabinoids CB1 receptors antagonists pain weight gain obesity LH-21 LH21 central