Arachidonic acid leelamide is the arachidonic amide analog of leelamine. Leelamine has weak affinity for the human CB1 and CB2 receptors, exhibiting 20% displacement of [3H]-CP55940 at a concentration of 10 μM.{14127} Leelamine inhibits PDK with an IC50 value of 9.5 μM.{14105} Derivatives of leelamine exhibit anti-inflammatory activity and show moderate inhibition of PLA2 activity from a variety of sources.{14107} There are no published studies of the pharmacological properties of arachidonic acid leelamide.
Size
5 mg
Concentration
n/a
Applications
n/a
Other Names
AA cannabinoids central peripheral CB1 CB2 CP55940 PDK pyruvates dehydrogenases kinases anti-inflammatory inflammation phospholipases PLA2 inhibits inhibitors inhibition cannabinoids cbs sythetic